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目錄號(hào)	產(chǎn)品名	產(chǎn)品描述	Selective / Pan	IC50 / Ki
S2894	SB742457	SB742457 (GSK 742457) is a highly selective 5-HT6 receptor antagonist with pKi of 9.63, exhibits >100-fold selectivity over other receptors. Phase 2.	Selective	5-HT6, pKi: 9.63
S2856	SB 271046 hydrochloride	SB 271046 hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pK_i of 8.9, exhibits 200-fold greater selectivity over other 5-HT receptor subtypes.	Selective	5-HT6, pKi: 8.92
S6087	Indophagolin	Indophagolin, a potent indoline-containing?autophagy?inhibitor with IC50 of 140 nM, antagonizes the purinergic receptor?P2X4?as well as P2X1?and P2X3?with IC50s of 2.71, 2.40 and 3.49 μM, respectively, also has a strong antagonistic effect on?serotonin receptor?5-HT6?with IC50 of 1.0 μM.	Selective	5-HT6, IC50: 1.0 μM
S1283	Asenapine maleate	Asenapine maleate (Org 5222) is a high-affinity antagonist of serotonin, norepinephrine, dopamine and histamine receptors, used for the treatment of schizophrenia and acute mania associated with?bipolar disorder.	Pan	5-HT6, pKi: 9.6
S3913	Pimethixene maleate	Pimethixene (Pimetixene) maleate, an antihistamine, anntimigraine agent and antiserotonergic compound, is a highly potent antagonist of a broad range of monoamine receptors, including a variety of serotonin receptors. Pimethixene maleate inhibits 5-HT2A, 5-HT2B, 5-HT2C, 5-HT1A, 5-HT1B, 5-HT6, 5-HT7, Adrenergic α-1A, Dopamine D1 Receptor, Dopamine D2 Receptor, Dopamine D4.4 Receptor, Histamine H1 Receptor, Muscarinic M1 and Muscarinic M2 with pKi of 10.22, 10.44, 8.42, 7.63, < 5, 7.	Pan	5-HT6, pKi: 7.30
S2677	BRL-15572 Dihydrochloride	BRL-15572 is a 5-HT1D receptor antagonist with pK_i of 7.9, also shows a considerable affinity at 5-HT1A and 5-HT2B receptors, exhibiting 60-fold selectivity over 5-HT1B receptor.	Pan	5-HT6, pKi: 5.9

5-HT6 選擇性抑制劑 | 拮抗劑